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[mr_b]

Nowość dostępna w UK.

What is Nifoxipam

Nifoxipam is a PAM ((positive allosteric modulator) of the benzodiazepine receptors, specifically the ‘diazepam sensitive’ sites. It has not been investigated but is a known to be a metabolite of flunitrazepam showing it has no toxic effects at the weights used for research.

What is Nifoxipam used for?

As an unexplored metabolite, a large range of in vivo and in-vitro research paths are open. The hydroxyl group may be esterified altering solubility values in different solvents. The hydroxyl may be deuterated and readily replaced by other groups giving a research compound with a VERY wide spectrum of uses.



IUPAC 5-(2-fluorophenyl)-3-hydroxy-7-nitro-1H-benzo[e][1,4]diazepin-2(3H)-one

CAS Number 74723-10-7

Molecular Formula C15H10F1O4N1

Molecular Weight 315.26

Formulation Crystalline solid

Purity ≥99%

Storage -20°C

Stability 2 years

SMILES O=C1C(O)N=C(C2=CC=CC=C2F)C3=CC([N+]([O-])=O)=CC=C3N1

LogP 10.45

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[Sierpień]

Z opisów na Bluelight wydaje się być dobre relaksująco nasenne benzo, aczkolwiek raczej słabe w działaniu. Jakieś info kiedy będzie dostępne w Polsce?